Pirenzepine Dihydrochloride

产品名称：

29868-97-1
Pirenzepine Dihydrochloride
5,11-Dihydro-11-[(4-methyl-1-piperazinyl)acetyl]-6H-pyrido[2,3-b][1,4]benzodiazepin-6-one Dihydrochloride

产品介绍：

产品说明

一般描述

Pirenzepine dihydrochloride is an anticholinergic agent. It is also considered as an antiulcer drug. It is used to treat myopia, gastric and duodenal ulcers. Pirenzepine dihydrochloride induces the dimerization of muscarinic M1 receptors.

应用

Pirenzepine dihydrochloride has been used

in transactivation of fibroblast growth factor receptor (FGFR).
as a supplement in cell culture.
for the stimulation of human fibroblasts

包装

500 mg in poly bottle
1 g in poly bottle

生化/生理作用

Selective M₁ muscarinic acetylcholine receptor antagonist.

特点和优势

This compound is a featured product for Neuroscience research. Click here to discover more featured Neuroscience products. Learn more about bioactive small molecules for other areas of research at sigma.com/discover-bsm.
This compound is featured on the Acetylcholine Receptors (Muscarinic) page of the Handbook of Receptor Classification and Signal Transduction. To browse other handbook pages, click here.

注意

Hygroscopic; store desiccated at room temperature.

基本信息

经验(实验)分子式	C₁₉H₂₁N₅O₂ · 2HCl
分子量	424.32
EC 号	249-907-5
MDL编号	MFCD00055214
PubChem化学物质编号	24277863
NACRES	NA.77

产品性质

质量水平	200
测定	≥98% (TLC)
形式	powder
颜色	white
溶解性	H₂O: 50 mg/mL
SMILES string	Cl[H].Cl[H].CN1CCN(CC1)CC(=O)N2c3ccccc3C(=O)Nc4cccnc24
InChI	1S/C19H21N5O2.2ClH/c1-22-9-11-23(12-10-22)13-17(25)24-16-7-3-2-5-14(16)19(26)21-15-6-4-8-20-18(15)24;;/h2-8H,9-13H2,1H3,(H,21,26);2*1H
InChI key	FFNMBRCFFADNAO-UHFFFAOYSA-N
Gene Information	human ... CHRM1(1128)

安全信息

储存分类代码	13 - Non Combustible Solids
WGK	WGK 2
闪点(F)	Not applicable
闪点(C)	Not applicable
个人防护装备	Eyeshields, Gloves, type N95 (US)