1,5-Dansyl-Glu-Gly-Arg Chloromethyl Ketone, Dihydrochloride-Calbiochem

产品说明

一般描述

Effective irreversible inhibitor of uPA, Factor Xa, and urokinase. Fluorophore allows direct monitoring of interactions of labeled enzyme. Does not inhibit tPA.

包装

5 mg in Plastic ampoule

生化/生理作用

Product does not compete with ATP.
Reversible: no
Target IC₅₀: 100 nM for factor Xa
Cell permeable: no
Primary Target
UPA

警告

Toxicity: Standard Handling (A)

重悬

Reconstitute at 1 mg/ml in 10 mM HCl. Dilute with physiological buffers just prior to use.
Following initial thaw, aliquot and refrigerate (4°C). Stock solutions are stable for up to 4 months at 4°C.

其他说明

Bajaj, S.P., et al. 1992. Proc. Natl. Acad. Sci. USA89, 152.
Bergmeyer, H.V. 1984. Methods Enzym. Anal. 5, 375.
Kettner, C., and Shaw, E. 1981. Methods Enzymol.80, 826.

法律信息

CALBIOCHEM is a registered trademark of Merck KGaA, Darmstadt, Germany

产品性质

安全信息