产品说明
包装
5, 25 mg in glass bottle
生化/生理作用
LY2033298 is a robust allosteric potentiator that is highly selective for the human M4 muscarinic acetylcholine receptor subtype. LY2033298 potentiates ACh-M4 binding, with no effect at M1/3/5 receptors. LY2033298 can also bind to the M ACh receptor, and mediate either positive or negative allosteric effects depending on the ligand used to probe receptor activity.
特点和优势
This compound was developed by Eli Lilly. To browse the list of other pharma-developed compounds and Approved Drugs/Drug Candidates, click here.
基本信息
| 经验(实验)分子式 | C13H14ClN3O2S |
| 分子量 | 311.79 |
| MDL编号 | MFCD12912423 |
| PubChem化学物质编号 | 329817677 |
| NACRES | NA.77 |
产品性质
| 质量水平 | 100 |
| 测定 | ≥98% (HPLC) |
| 形式 | solid |
| 储存条件 | desiccated |
| 颜色 | off-white to tan |
| 溶解性 | DMSO: >20 mg/mL |
| 创始人 | Eli Lilly |
| 储存温度 | −20℃ |
| SMILES string | COc1nc2sc(C(=O)NC3CC3)c(N)c2c(C)c1Cl |
| InChI | 1S/C13H14ClN3O2S/c1-5-7-9(15)10(11(18)16-6-3-4-6)20-13(7)17-12(19-2)8(5)14/h6H,3-4,15H2,1-2H3,(H,16,18) |
| InChI key | CTEGQKDJTBWFHW-UHFFFAOYSA-N |
安全信息
| 象形图 |  |
| 警示用语： | Danger |
| 危险声明 | H334 |
| 预防措施声明 | P261 - P284 - P501 |
| 危险分类 | Resp. Sens. 1 |
| 储存分类代码 | 11 - Combustible Solids |
| WGK | WGK 3 |
| 闪点(F) | Not applicable |
| 闪点(C) | Not applicable |
Sigma-Aldrich
m.cnreagent.com
