3,7-二甲基-1-炔丙基黄嘌呤

产品名称：

14114-46-6
3,7-Dimethyl-1-propargylxanthine
3,7-Dimethyl-1-(2-propynyl)xanthine
DMPX
3,7-二甲基-1-炔丙基黄嘌呤

产品介绍：

产品说明

应用

3,7-Dimethyl-1-propargylxanthine (DMPX) has been used as an A₂ -adenosine receptor (AR) antagonist:

to study its effects on potential modulation of motor output elicited by epidural spinal stimulation (ESS)
to study the role of A_2areceptor in elevating cyclic adenosine monophosphate (cAMP) levels
to study its effects on the cell viability of human gastric cancer cell line

包装

10, 25, 100 mg in poly bottle

生化/生理作用

3,7-Dimethyl-1-propargylxanthine (DMPX) is a caffeine analog and A₂-selective adenosine receptor (AR) antagonist.

基本信息

产品性质

质量水平	100
测定	≥98% (HPLC)
形式	powder
颜色	white to beige
溶解性	DMSO: 15 mg/mL, clear
SMILES string	CN1C(=O)N(CC#C)C(=O)c2c1ncn2C
InChI	1S/C10H10N4O2/c1-4-5-14-9(15)7-8(11-6-12(7)2)13(3)10(14)16/h1,6H,5H2,2-3H3
InChI key	IORPOFJLSIHJOG-UHFFFAOYSA-N
Gene Information	human ... ADORA2A(135), ADORA2B(136) rat ... Adora1(29290), Adora2a(25369)

安全信息

象形图
警示用语：	Warning
危险声明	H315 - H319 - H335
预防措施声明	P302 + P352 - P305 + P351 + P338
危险分类	Eye Irrit. 2 - Skin Irrit. 2 - STOT SE 3
靶器官	Respiratory system
储存分类代码	11 - Combustible Solids
WGK	WGK 3
个人防护装备	dust mask type N95 (US), Eyeshields, Gloves